Clenbuterol for weight loss. Instructions for use for women and men. How to take pills, courses, side effects. Reviews

Clenbuterol is a bronchodilator, the main purpose of which is to treat asthma and eliminate the symptoms of the disease. In bodybuilding and fitness, the drug has become widespread due to the powerful effect of the active substance on metabolic processes.

Clenbuterol for weight loss has been used for several decades and its effectiveness in burning fat has been confirmed by numerous studies.

Chemical composition and release form

Clenbuterol hydrochloride, according to the mechanism of action, is a selective β2-adrenostimulant. This compound is the main component of the "Clenbuterol" drug, which is available in tablets and syrup. Different forms of release differ in the concentration of the active substance.

Active ingredient content:

• in tablets - 0.02 mg;
• in syrup - 0.01 mg / 5 ml;
• children's syrup 0.001 mg / 5 ml.

Tablets are available in blister packs and glass bottles of 20, 50 and 100 pieces. The syrup is available in 50 ml bottles and has a limited shelf life due to its high sugar content.

How it helps in losing weight

The drug is not intended to reduce body weight, but has been successfully used in bodybuilding to reduce the volume of adipose tissue without destroying muscle fibers. At the level of professional sports, Clenbuterol was officially banned by WADA in 1992 as a pharmacological doping.

Clenbuterol for weight loss is effective due to its ability to regulate hormonal processes. The active ingredient triggers a series of sequential reactions that affect the biochemistry of the body. As a result of taking the drug, the activity of cells responsible for the transport and processing of lipids in the body increases.

The step-by-step mechanism of the effect of a substance on the human body is described below:

1. The active substance of the drug binds to β2-receptors in muscle and adipose tissue.
2. Receptors activate the production of cyclic adenosine monophosphate, a substance that is responsible for the transmission of hormonal signals between cells.
3. The result is the active production of enzymes that transport fatty acid molecules from fat cells to muscles, where they are converted into energy.

After 15 minutes, a high concentration of adrenaline, insulin and norepinephrine is observed in the blood of a person who has taken the drug. The hormonal surge in combination with the production of enzymes increases the rate of metabolic processes by 20-30%.

The main advantage of the drug for athletes is that it blocks catabolism, allowing you to eliminate excess fats without exerting a destructive effect on muscle fibers.

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Indications for use

Traditionally, clenbuterol is used by official medicine in the complex therapy of pathologies and diseases of the respiratory system.

Diagnoses for which reception is indicated:

• bronchial asthma;
• broncho-obstructive syndrome;
• COPD.

In bodybuilding and fitness, the drug is indicated for achieving the desired parameters of the percentage of adipose tissue and muscle, losing weight, improving endurance and increasing the effectiveness of training.

Athletes supplement the drug with a set of measures necessary to achieve a competitive form - drawing of muscle relief.

Contraindications

The risk of using the drug in the presence of contraindications is high. The use of even small doses can provoke a heart attack or lead to the development of a pre-infarction state.

The possibility of using clenbuterol for the following diseases and conditions is excluded:

• myocardial infarction;
• subaortic aortic stenosis;
• heart failure;
• tachyarrhythmia;
• tachycardia;
• endocrine disorders;
• pathology of the thyroid gland;
• allergic reaction.

For women at the stage of breastfeeding or pregnancy, the doctor determines the possibility of prescribing the drug. If the potential benefits outweigh the risks, the drug is prescribed with an individual selection of dosage.

Rules and recommendations for admission

Clenbuterol for weight loss or fat burning requires changes in diet and daily habits to prevent unwanted body reactions and neutralize toxic effects.

Below are the basic rules for admission:

1. It is safest to start taking it at 6-8 weeks of drying, when the metabolic rate has decreased as a result of the low content of fast carbohydrates.
2. Clenbuterol should be taken in the morning to avoid problems with falling asleep and sleep quality as a result of stimulating adrenaline production.
3. The duration of use is no more than 2 weeks. During this period, the body develops tolerance to the active substance, and further intake will give zero result.
4. For effectiveness, a daily dose increase is required up to 6 days.
5. The dosage cannot be increased on subsequent days.
6. Increasing the dosage is accompanied by a separate intake - in the morning and at lunchtime, to avoid overdose.
7. It is necessary to start a gradual dose reduction 2-3 days before the end of the course.
8. Strong coffee and alcohol are temporarily strictly prohibited. The combination of ethyl alcohol and caffeine with an active ingredient increases the risk of side effects and inhibits lipolysis (fat burning).
9. If the course of admission did not give the desired result, it can be safely repeated only after a break of 14 days.
10. The effectiveness of taking clenbuterol depends on the diet. Depending on your goals, you should follow a specialized diet low in simple carbohydrates and high in protein.
11. Increased aerobic loads are shown throughout the course.
12. When performing exercises of an aerobic nature, control of heart rate and blood pressure should be strengthened.

The appearance of symptoms of dysfunction of the heart ventricles, tingling and burning sensation in the region of the heart is a signal for immediate discontinuation of clenbuterol and a visit to the doctor.

Determining a safe dosage

In the absence of an underlying medical indication, there is no safe dosage. Experts in sports pharmacology have developed dosage regimens that maximize potential harm while maintaining effectiveness.

It is:

• for women - no more than 120 mcg per day;
• for men - no more than 140 mcg per day.

This is the maximum allowable daily amount, which is achieved on the sixth day of admission by increasing the dosage from 20 mcg.Taking the maximum dose on the first day can lead to the development of an attack of respiratory and heart failure.

Clenbuterol course without ketotifen

Self-administration of ketotifen without auxiliary medications cannot last longer than 14 days. In the third week, the receptors stop responding to the substance that has entered the body, and addiction develops. The reception scheme is presented in the table.

Clenbuterol + ketotifen course

The complex of ketotifen and clenbuterol can reduce the risk of side effects or reduce their severity. The use of a combination of two drugs allows you to extend the course time. Ketotifen is needed during a break to quickly restore receptor sensitivity.

Taking these drugs can be combined - this makes it possible to use clenbuterol for 4-8 weeks. The scheme for taking clenbuterol is the same as when taking the drug alone, but on day 5, in the evening, ketotifen is added at a dosage of 2 mg.

Clenbuterol + T3 + yohimbine course

Tetraiodothyronine (T3) is a drug that, in combination with clenbuterol and yohimbine, provides synergy. Sports drug manufacturers use this combination to create powerful, fast-acting stimulants and fat burners.

The duration of the course is 3 weeks. The dosage regimen involves increasing the dose every 3 days. From day 12, it is necessary to reduce the dose in the reverse order.

Side effects

Taking clenbuterol for weight loss is fraught with side effects even in the absence of contraindications.

Below is a list of side effects from the drug:

• heart palpitations occur in 60% of people taking the drug. Eliminated with adrenergic blocking drugs;
• tremors, tremors and weakness. It takes place on the 2-3 day of admission;
• increased sweating;
• sleep disturbances, insomnia;
• anxiety, panic attacks. It is eliminated after taking ketotifen;
• instability of blood pressure. You can prevent and eliminate with the help of adrenergic blockers;
• nausea and diarrhea;
• convulsions.

Most of the side effects can be eliminated by accompanying the intake of clenbuterol with ketotifen and adrenergic blocking drugs. In case of an overdose, side effects will become more pronounced, in addition, toxic damage to the myocardium and the male reproductive system is possible.

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Interaction with other drugs

At the time of taking clenbuterol, you should stop taking medications, as this increases the risk of side effects and toxic effects.

Below are the drugs and substances with which clenbuterol is incompatible:

• ephedrine and its synthetic analogues in combination with clenbuterol increase the risk of developing heart disease as a result of taking;
• in combination with cardiac glycosides, the drug causes a violation of the heart rhythm;
• impairs the effectiveness of hypoglycemic drugs;
• theophylline enhances the destructive effect on the heart muscle.

Clenbuterol for weight loss is often combined with drug synergists - anabolic steroids.

Strengthening the effectiveness of the drug, they simultaneously increase the risk of developing cardiac muscle hypertrophy. Simultaneous reception is possible no longer than 3 days at the end of the course.

Where to buy, price, release forms

Clenbuterol from various pharmaceutical companies is present in the range of pharmacies. The complexity of the acquisition lies in the fact that this pharmacological drug is included in the category of prescription drugs.In the absence of a prescription, you can buy the drug at any sports pharmacology store.

The cost of clenbuterol depends on the country of origin, the form of release and the concentration of the active ingredient. The average drug cost in dollar terms is described in the table below.

Storage conditions and shelf life

The drug Clenbuterol does not require special storage conditions. The tablets should be stored in a dry place where the air temperature does not exceed 25 degrees. The shelf life of the drug is 3 years from the date of manufacture. For syrup, the maximum shelf life is 2 years from the date of production, but no more than 30 days from the moment the bottle is opened. Store the syrup in a cool, dark place.

Studies on weight loss with Clenbuterol

The first scientific confirmation of the effectiveness of clenbuterol in weight loss was provided in 2015 by Australian scientists from the Garvan Institute for Medical Research. Scientists have investigated the effect of a similar substance, formoterol, given a daily dose of 160 mcg.

As a result of research, it was found that taking the drug in a course leads to the following results:

• anabolism is activated;
• protein synthesis is stimulated.

Combined with the stimulation of adrenaline production, these effects make it possible to lose weight by reducing the volume of adipose tissue and preserving muscle. The author of the book "Anabolic Steroids" Leonid Ostapenko described in detail the mechanism of the development of side effects with the regular use of clenbuterol to eliminate excess adipose tissue.

According to the research conducted by the author, the clenbuterol molecule tends to accumulate in the cells of organs, gradually provoking their pathological growth. Due to the abuse of the drug, hypertrophy of the internal organs occurs, and favorable conditions are created for the growth of malignant neoplasms.

How Clenbuterol affects the heart

The consequence of taking the drug is a destructive effect on the functioning of the cardiovascular system.

Stimulating the production of adrenaline provokes:

• increased heart rate;
• vascular spasms;
• increased blood pressure.

The use of the drug leads to the depletion of potassium and magnesium reserves, which affects the condition of the heart muscle. Asparkam and ketotifen eliminate both problems. If, after supplementing the course with these drugs, heart problems have not been eliminated, you should cancel the appointment and undergo a cardiological examination.

Effects on sleep

As a result of research, it was found that 8% of people taking clenbuterol faced the problem of sleep disturbance. Insomnia, frequent nocturnal awakenings are the result of overstimulation of the nervous system.

The half-life of the drug from the human body is 24-26 hours. This means that the maximum concentration of the stimulating substance remains in the body throughout the day. To achieve significant results in weight loss, this feature of the drug is an advantage.

But, this feature is the cause of frequent sleep disorders. Side effects are neutralized with ketotifen. If sleep disorders are systematic and do not stop even with the accompanying evening intake of ketotifen, weight loss should be continued without clenbuterol or take a temporary break.

Clenbuterol depletes potassium stores

Clenbuterol for weight loss is combined with a specialized diet high in protein and potassium. The protein component is necessary to maintain muscle tissue volumes, activate ketabolism. Potassium is necessary to compensate for the deficiency of this element caused by taking clenbuterol.

As a result of stimulation of β2-adrenergic receptors in the kidneys with clenbuterol, renin production is increased. The consequence of this process is the leaching of potassium from the body, and its deficiency leads to a violation of the water-salt balance and other negative consequences for the body.

Potassium deficiency symptoms:

• trouble concentrating;
• decline in intellectual abilities;
• brittle hair;
• dry skin;
• muscle weakness;
• violation of the heart rhythm;
• increased fatigue;
• headaches;
• increased blood pressure;
• disorder of urination;
• diseases of the digestive system;
• violation of the functioning of the reproductive system.

There are several ways to prevent potassium deficiency while taking clenbuterol for weight loss:

1. Inclusion in the diet of foods rich in this substance.
2. The use of mineral supplements.
3. Taking medications to correct potassium deficiency.

Subject to the rules of admission and the duration of the course, potassium deficiency can be avoided by enhancing the diet with products that supply compounds of this substance to the body.

Doctors' Opinions on Safety and Efficacy: Should You Take?

The opinions of doctors regarding the use of clenbuterol in sports are divided. Science confirms the effectiveness of the drug as a fat burner, but warns against abuse. Doctors say that only absolutely healthy people can use the drug. It is recommended to be examined by a cardiologist and endocrinologist to avoid negative consequences.

Clenbuterol for weight loss is not a panacea, but only enhances the result of training and sports diet. It is impossible to achieve significant results in burning fat without normalizing nutrition and aerobic training.

Author: alexvasilena

Article design: Oksana Grivina

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